Palladium-catalyzed ortho-C-H alkenylation of 2-benzyl-1,2,3-triazoles.

نویسندگان

  • Ping He
  • Qingshan Tian
  • Chunxiang Kuang
چکیده

A mild and efficient method for the direct alkenylation of 2-benzyl-1,2,3-triazoles via Pd-catalyzed C-H bond activation was developed. This protocol was compatible with various substrates and gave the corresponding products in good to excellent yields. Thus, the present study provides a novel and valuable method for the synthesis of 2-benzyl-1,2,3-triazole derivatives.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 13 26  شماره 

صفحات  -

تاریخ انتشار 2015